May 2011 USANs


The May 2011 USANs have been published.

USAN Research Code StructureDrug Type Drug Class Target
alisertib, alisertib sodiumMLN-8237synthetic small moleculetherapeuticAURa, AURb
asunaprevirBMS-650032synthetic small moleculetherapeuticHCV NS3
cariprazine, cariprazine hydrochlorideRGH-188synthetic small moleculetherapeuticD2R D3R
ceftolozane, ceftolozane sulfateCXA-101natural product-derived small moleculetherapeuticvarious PBPs
crenezumabMABT5102Amonoclonal antibodytherapeuticAbeta
dalanterceptACE-041proteintherapeuticTGFbeta family
delcasertib, delcasertib acetateKAI-9803, BMS-875944peptidetherapeuticPKCdelta
epelsiban, epelsiban besylateGSK-557296Bsynthetic small moleculetherapeuticOxytocin receptor
erismodegibLDE-225synthetic small moleculetherapeuticSmo
evacetrapibLY-2484595synthetic small moleculetherapeuticCETP
ficlatuzumabSCH-900105, AV-299monoclonal antibodytherapeuticHGF
galeteroneTOK-001, VN-124natural product-derived small moleculetherapeuticAR
icopasent ethylAMR-101natural product-derived small moleculesupplement-
macitentanACT-064992synthetic small moleculetherapeuticETRa ETRb
oclacitinib, oclacitinib maleatePF-03394197synthetic small moleculetherapeutic
sarilumabREG-N88, SAR-153191monoclonal antibodytherapeuticIL6R
sitaxentan sodiumTBC-11251z, TBC-11251Nasynthetic small moleculetherapeuticETRa ETRb
tofacitinib citrateCP-690550-10synthetic small moleculetherapeuticJAK2, JAK3
trametinib, trametinib dimethyl sulfoxideGSK-1120212synthetic small moleculetherapeuticMEK
volasertib, volasertib trihydrochlorideBI-6727synthetic small moleculetherapeuticPLK1
vonicog alfaBAX-111proteinsupplement

A fair few kinase inhibitors, but does anyone know anything about Oclacitinib - Google shows only some dog cancer trials at the moment?