| USAN | Research Code | InChIKey (Parent) | Drug Class | Therapeutic class | Target |
| avarofloxacin hydrochloride | JNJ-32729463 | UAJMNUKJPPPJJT-CLNHMMGSSA-N | synthetic small molecule | therapeutic | topo II |
| lubabegron, lubabegron fumarate | LY-488756 | WIKLBKJBYSBYLL-QHCPKHFHSA-N | synthetic small molecule | therapeutic | beta 3 receptor |
| methylsamidorphan chloride | RDC-1036-03 | | natural product-derived small molecule | therapeutic | opioid receptors |
| palbociclib isethionate | PD-332991, PF-00080665 | AHJRHEGDXFFMBM-UHFFFAOYSA-N | synthetic small molecule | therapeutic | CDK4 CDK6 |
| pevonedistat hydrochloride | MLN-4924 | UPOLJMQMGITQAT-MNDZRTMASA-N | synthetic small molecule | therapeutic | NAE |
| rivipansel sodium | GMI-1070, PF-06460031 | | natural product-derived small molecule | therapeutic | selectins |
| sarecycline, sarecycline hydrochloride | P-005672 | APPRLAGZQKOUFL-UHFFFAOYSA-N | natural product derived small molecule | therapeutic | 30S ribosome |
| tenofovir alafenamide fumarate | GS-7340 | LDEKQSIMHVQZJK-CAQYMETFSA-N | synthetic small molecule | therapeutic prodrug | HIV RT |
| velcalcetide | KAI-4169 | C.dCdAdRdRdRdAdR | peptide | therapeutic | CaSr |
