May 2011 USANs
The May 2011 USANs have been published.
USAN | Research Code | Structure | Drug Type | Drug Class | Target |
alisertib, alisertib sodium | MLN-8237 | ![]() | synthetic small molecule | therapeutic | AURa, AURb |
asunaprevir | BMS-650032 | ![]() | synthetic small molecule | therapeutic | HCV NS3 |
cariprazine, cariprazine hydrochloride | RGH-188 | ![]() | synthetic small molecule | therapeutic | D2R D3R |
ceftolozane, ceftolozane sulfate | CXA-101 | ![]() | natural product-derived small molecule | therapeutic | various PBPs |
crenezumab | MABT5102A | monoclonal antibody | therapeutic | Abeta | |
dalantercept | ACE-041 | ![]() | protein | therapeutic | TGFbeta family |
delcasertib, delcasertib acetate | KAI-9803, BMS-875944 | ![]() | peptide | therapeutic | PKCdelta |
epelsiban, epelsiban besylate | GSK-557296B | ![]() | synthetic small molecule | therapeutic | Oxytocin receptor |
erismodegib | LDE-225 | ![]() | synthetic small molecule | therapeutic | Smo |
evacetrapib | LY-2484595 | ![]() | synthetic small molecule | therapeutic | CETP |
ficlatuzumab | SCH-900105, AV-299 | monoclonal antibody | therapeutic | HGF | |
galeterone | TOK-001, VN-124 | ![]() | natural product-derived small molecule | therapeutic | AR |
icopasent ethyl | AMR-101 | ![]() | natural product-derived small molecule | supplement | - |
macitentan | ACT-064992 | ![]() | synthetic small molecule | therapeutic | ETRa ETRb |
oclacitinib, oclacitinib maleate | PF-03394197 | ![]() | synthetic small molecule | therapeutic | |
sarilumab | REG-N88, SAR-153191 | monoclonal antibody | therapeutic | IL6R | |
sitaxentan sodium | TBC-11251z, TBC-11251Na | ![]() | synthetic small molecule | therapeutic | ETRa ETRb |
tofacitinib citrate | CP-690550-10 | ![]() | synthetic small molecule | therapeutic | JAK2, JAK3 |
trametinib, trametinib dimethyl sulfoxide | GSK-1120212 | ![]() | synthetic small molecule | therapeutic | MEK |
volasertib, volasertib trihydrochloride | BI-6727 | ![]() | synthetic small molecule | therapeutic | PLK1 |
vonicog alfa | BAX-111 | ![]() | protein | supplement |
A fair few kinase inhibitors, but does anyone know anything about Oclacitinib - Google shows only some dog cancer trials at the moment?